2008: COSMOtherm & COSMO-RS publications                      Return to Index


Prediction of partition coefficients using COSMO-RS: Solvent screening for maximum conversion in biocatalytic two-phase reaction systems
AC Spieß, W Eberhard, M Peters, MF Eckstein, L Greiner & J Büchs;  Chem Eng & Proc: Process Intensification, Volume 47, Issue 6, June 2008, Pages 1034-1041
DOI: 10.1016/j.cep.2007.02.007

COSMO-RS predicted the correct trends for the partition coefficients of solutes in different solvents. The calculated overall reaction equilibrium using these partition coefficients resulted in the prediction of the correct best solvent regarding conversion.


Structures of ionic liquids dictate the conversion and selectivity of enzymatic glycerolysis: theoretical characterization by COSMO-RS.
Chen B, Guo Z, Tan T, Xu X; Biotechnol Bioeng. 2008 Jan 1;99(1):18-29.

Using COSMO-RS calculations, this is the first attempt to characterize the IL structure-dependency of reaction specificity by associating structural variations of ILs with thermodynamic property changes of dissolved compounds and subsequent effects on reaction specificity.


On the miscibility of ethers and perfluorocarbons An experimental and theoretical study
P Babiak, A Nemcová, L Rulíšek, P Beier; Journal of Fluorine Chemistry, Vol 129, Issue 5, May 2008, Pages 397-401

Theoretical calculations of the miscibility temperatures of organic solvents and perfluorocarbons using COSMO-RS method were correlated with experimental data. Considering the difficulties in the accurate description of the macroscopic properties, such as miscibility temperatures, from the first principles, the agreement between experimental and theoretical data is reasonable.


Prediction of physicochemical properties of energetic materials
RK Toghiani, H Toghiani, SW Maloney and VM Boddu; Fluid Phase Equilibria, Vol 264, Issues 1-2, 1 March 2008, Pages 86-92
DOI: 10.1016/j.fluid.2007.10.018

The physicochemical properties of six new materials under consideration as munitions is estimated using COSMO-RS and group contribution methods, in order to asses their potential environmental fate before committing to full development.


Mutual Solubilities of Water and the [Cnmim][Tf2N] Hydrophobic Ionic Liquids
MG Freire, PJ Carvalho, RL Gardas, IM Marrucho, LMNBF Santos, and JAP Coutinho; J. Phys. Chem. B, 112 (6), 1604 -1610, 2008.
DOI: 10.1021/jp7097203 S1520-6106(70)09720-1

The predictive capability of COSMO-RS was evaluated for the description of the ionic liquid binary systems investigated. Acceptable agreement was found between the COSMO-RS predictions and the experimental data, both with the temperature dependence and with the ILs structural variations.


Partition Behavior of Hexachlorocyclohexane Isomers
K Goss, HPH Arp, G Bronner, C Niederer; J. Chem. Eng. Data, 53 (3), 750–754, 2008.
DOI: 10.1021/je700595y

The properties of the alpha, beta and gamma isomers of hexachlorocyclohexane were measured and compared with calculated results. SPARC and EPI-suite failed to predict any isomeric differences, however, COSMOtherm correctly predicted the qualitative differences between the isomers.


Quality control for plant metabolomics: reporting MSI-compliant studies
O Fiehn, G Wohlgemuth, M Scholz, T Kind, DY Lee, Y Lu, S Moon, B Nikolau (2008) Quality control for plant metabolomics: reporting MSI-compliant studies, The Plant Journal 53 (4) , 691–704
DOI: 10.1111/j.1365-313X.2007.03387.x

COSMO-RS and COSMOfrag were used for the rational design of solvent extractions mixtures for biologically active compounds.  A ternary mixture of methanol:chloroform:water (3:1:1) was predicted to dissolve a wider range of compounds than any single solvent, and verified experimentally.


Improvement of bioavailability of water insoluble drugs: Estimation of intrinsic bioavailability
J Kim, DH Jung, H Rhee, SH Choi, MJ Sung, WS Choi, Korean Journal of Chemical Engineering, Volume 25, No. 1, January, 2008, Pages 171-175, (Springer New York)
DOI: 10.1007/s11814-008-0031-4

The solubility of UDCA is seriously underpredicted both by the Syracuse function and Cerius 2. However, the COSMOtherm implementation of the COSMO-RS method provides a prediction close to the experimental measurement.


Effect of ortho-chlorine substitution on the partition behavior of chlorophenols.
C Neider, KU Goss,  Chemosphere. 2008 Mar;71(4):697-702. Epub 2008 Feb 20

The position of the chlorine substituent in chlorophenols is known to have a marked effect on the octanol/water and octane/water partition constants.  QSAR methods, including SPARC, failed to correctly predict the influence.  Only COSMOtherm, was shown to correctly reproduce these effects.


The pKa Values of PFOA and Other Highly Fluorinated Carboxylic Acids
KU Goss, Environ. Sci. Technol., 42 (2), 456–458, 2008. 10.1021/es702192c

Both COSMOtherm and SPARC were used to estimate pKa of environmentally important PFOAs.  While the presented work could not provide the exact experimental values for PFOA and other acids, it probably provides the most reasonable numbers that are available so far.